
[Dmt1]DALDA analogues with enhanced μ opioid agonist potency and with a mixed μ/κ opioid activity profile
Keywords: Boc; tert-butyloxycarbonyl; DAMGO; H-Tyr-d-Ala-Gly-Phe(NMe)-Gly-ol; Dmp; 2â²,6â²-dimethylphenylalanine; Dmt; 2â²,6â²-dimethyltyrosine; [Dmt1]DALDA; H-Dmt-d-Arg-Phe-Lys-NH2; DSLET; H-Tyr-d-Ser-Gly-Phe-Leu-Thr-OH; EDT; 1,2-ethanediol; Emp; 2â²-ethyl-6â